2,6-二氯-N,N-二乙基-4-氨基嘧啶合成路线 (共 2 条)
反应条件
triethylamine in ethanol
T=0°C; 0.5 h;
参考文献
SYNTA PHARMACEUTICALS CORP.
Patent: WO2006/53109 A1, 2006 ;
Location in patent: Page/Page column 99-100 ;
反应条件
sodium hydride in N,N-dimethyl-formamide
0.333333 h; Ambient temperature;
参考文献
Botta; Saladino; Anzini; Corelli
Nucleosides and Nucleotides, 1994 , vol. 13, # 8 p. 1769 - 1777