反应条件
1: 77 percent / various solvent(s) / 1 h / 230 - 240 °C
2: 1.) NaH / 1.) DMF, RT, 5 min, 2.) DMF, RT, overnight
View Scheme
参考文献
Musser, John H.; Brown, Richard E.; Loev, Bernard; Bailey, Kevin; Jones, Howard; et al.
Journal of Medicinal Chemistry, 1984 , vol. 27, # 2 p. 121 - 125