1: chloroacetic acid With dicyclohexyl-carbodiimide in dichloromethane T=20°C; 0.5 h; 2: n-dipropylamine With 4-(N,N-dimethlyamino)pyridine in dichloromethane T=20°C;
参考文献
Falco, Jose Luis; Pique, Maria; Gonzalez, Miguel; Buira, Irma; Mendez, Eva; Terencio, Jose; Perez, Cristina; Princep, Marta; Palomer, Albert; Guglietta, Antonio
European Journal of Medicinal Chemistry, 2006 , vol. 41, # 8 p. 985 - 990