反应条件
N,N,N',N',N'',N''-hexamethylphosphoric triamide; lithium diisopropyl amide 1.) THF, hexane, 50 deg C, 2 h, 2.) THF, hexane, 25 deg C, 2 h; Yield given. Multistep reaction;
参考文献
Labaudiniere, Richard; Hilboll, Gerd; Leon-Lomeli, Alicia; Terlain, Bernard; Cavy, Francoise; et al.
Journal of Medicinal Chemistry, 1992 , vol. 35, # 17 p. 3170 - 3179