1-BOC-4-(3-溴苯氧基)哌啶合成路线 （共 3 条）
反应条件
caesium carbonate in N,N-dimethyl-formamide T=65°C; 14 h;
参考文献
AURIGENE DISCOVERY TECHNOLOGIES LIMITED; UM PHARMAUJI SDN. BHD; GUMMADI, Venkateshwar, Rao; HOSAHALLI, Subramanya; NANDURI, Srinivas; AGGUNDA RENUKAPPA, Girish
Patent: WO2014/6554 A1, 2014 ;
Location in patent: Page/Page column 43; 44 ;
反应条件
potassium carbonate in N,N-dimethyl-formamide T=80°C; 16 h;
参考文献
Sato, Kenjiro; Sugimoto, Hiromichi; Rikimaru, Kentaro; Imoto, Hiroshi; Kamaura, Masahiro; Negoro, Nobuyuki; Tsujihata, Yoshiyuki; Miyashita, Hirohisa; Odani, Tomoyuki; Murata, Toshiki
Bioorganic and Medicinal Chemistry, 2014 , vol. 22, # 5 p. 1649 - 1666
反应条件
triphenylphosphine; diethylazodicarboxylate in tetrahydrofuran T=0°C; Inert atmosphere;
参考文献
KADMON CORPORATION, LLC; BOXER, Michael; RYAN, John; TONRA, James
Patent: WO2014/55999 A2, 2014 ;
Location in patent: Paragraph 0238 ;
