1: With N-ethyl-N,N-diisopropylamine; isobutyl chloroformate in tetrahydrofuran T=-10°C; 0.25 h; 2: With sodium tetrahydroborate; water in tetrahydrofuran T=-10°C; 0.0833333 h; Inert atmosphere;
参考文献
Rotstein, Benjamin H.; Yudin, Andrei K.
Synthesis (Germany), 2012 , vol. 44, # 18 p. 2851 - 2858