1: 1-(4-methoxybenzyl)-3,4-dihydroquinolin-2(1H)-one With lithium hexamethyldisilazane in tetrahydrofuran
T=-78°C; 0.5 h;
2: methyl iodide in tetrahydrofuran
参考文献
ELI LILLY AND COMPANY
Patent: WO2005/20975 A2, 2005 ;
Location in patent: Page/Page column 209 ;
WO 2005/020975 A2