反应条件
1: 4-benzyloxy-1H-indole With sodium hydride in N,N-dimethyl-formamide T=0°C; 0.0833333 h; 2: benzenesulfonyl chloride in N,N-dimethyl-formamide T=20°C; 0.5 h;
参考文献
Smart, Brian P.; Oslund, Rob C.; Walsh, Laura A.; Gelb, Michael H.
Journal of Medicinal Chemistry, 2006 , vol. 49, # 10 p. 2858 - 2860