反应条件
1: 1.) NaH / 1.) DMF, from RT to 70 deg C, 2.) DMF, 70 deg C, 2 h 2: 2.3 g / H2 / 10percent Pd/C / ethanol / 760 Torr View Scheme
参考文献
Closse, Annemarie; Haefliger, Walter; Hauser, Daniel; Gubler, Hans Ulrich; Dewald, Beatrice; Baggiolini, Marco
Journal of Medicinal Chemistry, 1981 , vol. 24, # 12 p. 1465 - 1471