1: With lithium hydroxide; water in methanol
T=90°C; 1.5 h;
2: With hydrogenchloride in 1,4-dioxane; water
T=100°C; 2 h;
3: With sodium carbonate in water
pH=8;
参考文献
PFIZER LIMITED
Patent: WO2008/135830 A1, 2008 ;
Location in patent: Page/Page column 61 ;
WO 2008/135830 A1