5-氯-3-(三氟甲基)吡啶-2-胺合成路线 (共 1 条)
反应条件
N-chloro-succinimide in N,N-dimethyl-formamide
T=60°C; 1 h;
参考文献
GLAXOSMITHKLINE LLC; BANKA, Anna; CATALANO, John, G.; CHONG, Pek, Yoke; FANG, Jing; GARRIDO, Dulce, Maria; PEAT, Andrew, James; PRICE, Daniel, J.; SHOTWELL, John, Brad; TAI, Vincent; ZHANG, Huichang
Patent: WO2011/41713 A2, 2011 ;
Location in patent: Page/Page column 206 ;