1-(4-苄氧基-3-氯苯基)哌嗪合成路线 (共 1 条)
反应条件
sodium t-butanolate; tris-(dibenzylideneacetone)dipalladium(0); 2,2'-bis-(diphenylphosphino)-1,1'- binaphthyl in toluene
T=110°C; 14 h;
参考文献
EXELIXIS, INC.
Patent: WO2005/117909 A2, 2005 ;
Location in patent: Page/Page column 102 ;
WO 2005/117909 A2