2-[2-氧代-2-(3-吡啶)乙基]-1H-异吲哚-1,3(2H)-二酮合成路线 (共 2 条)
反应条件
in DMF (N,N-dimethyl-formamide)
T=20°C; 72 h;
参考文献
OSI PHARMACEUTICALS, INC.
Patent: WO2004/104001 A2, 2004 ;
Location in patent: Page 66-67 ;
WO 2004/104001 A2
反应条件
sodium tetrahydroborate in water; isopropyl alcohol
T=20°C; 12 h;
参考文献
PROSIDION LIMITED
Patent: WO2006/56815 A1, 2006 ;
Location in patent: Page/Page column 18 ;