反应条件
1: 1.8 g / KOH, pyridine / pyridine / 3 h
2: 1.5 g / fused sodium acetate, glacial acetic acid / 4 h / Heating
3: H2 / 10percent Pd/C
View Scheme
参考文献
Oshitari, Tetsuta; Okuyama, Yuji; Miyata, Yoshiki; Kosano, Hiroshi; Takahashi, Hideyo; Natsugari, Hideaki
Bioorganic and Medicinal Chemistry Letters, 2011 , vol. 21, # 15 p. 4540 - 4544