反应条件
<b>Multi-step reaction with 3 steps<br /> </b>1.1: sodium hydride / N,N-dimethyl-formamide; mineral oil / 0.5 h / 0 °C<br />1.2: 24 h / 20 °C<br />2.1: acetic acid; sulfuric acid / 24 h / 90 - 95 °C<br />3.1: pyridine / 1 h / 20 °C<br /> <br />
参考文献
Jesus, Ana R.; Dias, Catarina; Matos, Ana M.; De Almeida, Rodrigo F.M.; Viana, Ana S.; Marcelo, Filipa; Ribeiro, Rogrio T.; Macedo, Maria P.; Airoldi, Cristina; Nicotra, Francesco; Martins, Alice; Cabrita, Eurico J.; Jimnez-Barbero, Jess; Rauter, Amlia P. Journal of Medicinal Chemistry, 2014 , vol. 57, # 22 p. 9463 - 9472