反应条件
caesium carbonate; tris-(dibenzylideneacetone)dipalladium(0); 9,9-dimethyl-4,5-bis(diphenyl-phosphino)xanthene in 1,4-dioxane
T=100°C; 16 h; Inert atmosphereSealed tube;
参考文献
PFIZER INC.; ARHANCET, Graciela Barbieri; CASIMIRO-GARCIA, Agustin; CHEN, Xiangyang; HEPWORTH, David; MEYERS, Marvin Jay; PIOTROWSKI, David Walter; RAHEJA, Raj Kumar
Patent: WO2010/116282 A1, 2010 ;
Location in patent: Page/Page column 63-64 ;
WO 2010/116282 A1