反应条件
1: 78 percent / ammoniac / methanol / 16 h / 120 °C / autoclave
2: 50 percent / hydroxide de potassium, brome / H2O / 1.) 0 deg C, 15 min, 2.) 80 deg C, 10 min.
3: 80 percent / acide chlorhydrique 12 N / H2O / 0.25 h
View Scheme
参考文献
Turck, Alain; Brument, Jean-Francois; Queguiner, Guy
Journal of Heterocyclic Chemistry, 1981 , vol. 18, p. 1465 - 1468