反应条件
1: 71 percent / 48percent HBr / acetic acid / 12 h / Heating
2: H2, aq. HCl / 10percent Pd/C / ethanol / 96 h / Ambient temperature
3: 55 percent / NaHCO3 / dimethylformamide / 4 h / Heating
View Scheme
参考文献
Dammertz; Reimann
Archiv der Pharmazie, 1982 , vol. 315, # 1 p. 27 - 32