反应条件
1: 4-(trifluoromethyl)phenol With sodium hydride in N,N-dimethyl-formamide
T=20°C; 0.5 h;
2: 1-bromo-3-chloro-1-phenylpropane in N,N-dimethyl-formamide
T=20°C; 60 h;
参考文献
Silvestri, Romano; Artico, Marino; La Regina, Giuseppe; Di Pasquali, Alessandra; De Martino, Gabriella; D'Auria, Felicia Diodata; Nencioni, Lucia; Palamara, Anna Teresa
Journal of Medicinal Chemistry, 2004 , vol. 47, # 16 p. 3924 - 3926