反应条件
1: Et3N / tetrahydrofuran / 0.25 h / 5 °C 2: tetrahydrofuran / Ambient temperature 3: 68 percent / H2, 10percent ethanolic NH3 / Rh/C / 80 °C / 43440.4 Torr 4: 66 percent / 3-methyl-butan-1-ol / 12 h / Heating View Scheme
参考文献
Journal of Medicinal Chemistry, , vol. 29, # 1 p. 19 - 25