反应条件
1: p-toluenesulfonic acid / ethane-1,2-diol / 72 h / Heating
2: 1.) n-BuLi / 1.) THF, hexane, 50 deg C, 3 h, 2.) THF, hexane, 50 deg C, 6 h
View Scheme
参考文献
Houlihan, William J.; Boja, John W.; Parrino, Vincent A.; Kopajtic, Theresa A.; Kuhar, Michael J.
Journal of Medicinal Chemistry, 1996 , vol. 39, # 25 p. 4935 - 4941