1-甲基-1H-1,2,4-噻唑-3-羧酸合成路线 (共 1 条)
反应条件
1: With water; potassium hydroxide in methanol
T=20°C; 3 h;
2: With acetic acid in methanol; N,N-dimethyl-formamide
参考文献
GLAXO GROUP LIMITED
Patent: WO2009/147188 A1, 2009 ;
Location in patent: Page/Page column 102 ;
WO 2009/147188 A1