1: K2CO3 / acetone; dimethylformamide; H2O / 18 h / Heating 2: HOAc, H2 / 10percent Pd/C / 20 h / 50 °C / 2585.7 Torr View Scheme
参考文献
DeMarinis, Robert M.; Gallagher, Gregory; Hall, Ralph F.; Franz, Robert G.; Webster, Charles; et al.
Journal of Medicinal Chemistry, 1986 , vol. 29, # 6 p. 939 - 947