1: 52.1 percent / formic acid / H2O / 48 h / 60 - 70 °C
2: 88.7 percent / triethylamine / CH2Cl2 / 20 °C
3: 37 percent / tin(IV) chloride / acetonitrile / 4 h / 50 - 55 °C
View Scheme
参考文献
Clark, Jeremy L.; Mason, J. Christian; Hobbs, Ann J.; Hollecker, Laurent; Schinazi, Raymond F.
Journal of Carbohydrate Chemistry, 2006 , vol. 25, # 6 p. 461 - 470