反应条件
1: 5-methyl-1H-indole With ethylmagnesium bromide in tetrahydrofuran
T=-78°C; 0.133333 - 0.166667 h;
2: 2-nitrobenzoic acid chloride in tetrahydrofuran
T=-78 - 20°C; 4.16667 h;
3: With hydrogenchloride; methanol; lithium hydroxide
more than 3 stages;