1: With lithium aluminium tetrahydride in tetrahydrofuran; diethyl ether T=20 - 45°C; 2: With sodium sulfate in tetrahydrofuran; diethyl ether 0.5 h; 3: With ammonium chloride in tetrahydrofuran; diethyl ether; water 0.25 h;
参考文献
Bristol Myers Squibb Company
Patent: US6982265 B1, 2006 ;
Location in patent: Page/Page column 29 ;
Mikhalitsyna, Elena A.; Tyurin, Vladimir S.; Nefedov, Sergey E.; Syrbu, Sergey A.; Semeikin, Aleksandr S.; Koifman, Oskar I.; Beletskaya, Irina P.
European Journal of Inorganic Chemistry, 2012 , # 36 p. 5979 - 5990