反应条件
1: 1.) n-butyllithium / 1.) ether, 20 deg C, 18 h, 2.) ether
2: 47 percent / aq. H2SO4 / 1 h / 115 °C
View Scheme
参考文献
Burke, Terrence R.; Jacobson, Arthur E.; Rice, Kenner C.; Weissman, Ben Avi; Huang, Hsueh-Cheng; Silverton, J. V.
Journal of Medicinal Chemistry, 1986 , vol. 29, # 5 p. 748 - 751