7,8-二氟-2,3-二氢-3-甲基-4-氢恶嗪合成路线 (共 11 条)
反应条件
1: 1 h / 140 - 145 °C 2: PPE / 1 h / 140 - 145 °C 3: 94 percent / conc. HCl / acetic acid / 3 h / Heating 4: 38 percent / dimethylsulfoxide / 1 h / 100 - 140 °C View Scheme
参考文献
Hayakawa; Hiramitsu; Tanaka
Chemical and Pharmaceutical Bulletin, 1984 , vol. 32, # 12 p. 4907 - 4913