N-[1-(S)-乙氧羰基-3-苯丙基]-L-丙氨酸合成路线 （共 47 条）
反应条件
1: 30.1 percent / K2CO3 / dimethylsulfoxide / 30 h / Ambient temperature 2: ethyl acetate; diisopropyl ether 3: 96 percent / H2 / Pd / ethanol / 3 h / 760 Torr / Ambient temperature View Scheme
参考文献
Journal of Medicinal Chemistry, , vol. 32, # 2 p. 289 - 297
反应条件
1: 43.6 percent / K2CO3 / dimethylsulfoxide / 30 h / Ambient temperature 2: ethyl acetate; diisopropyl ether 3: 96 percent / H2 / Pd / ethanol / 3 h / 760 Torr / Ambient temperature View Scheme
参考文献
Journal of Medicinal Chemistry, , vol. 32, # 2 p. 289 - 297
反应条件
in water; potassium carbonate; acetonitrile
反应条件
trifluoroacetic acid 2 h; Ambient temperature;
参考文献
Iwasaki; Kimura; Numao; Kondo
Chemical and Pharmaceutical Bulletin, 1989 , vol. 37, # 2 p. 280 - 283
反应条件
1: 77 percent / N(C2H5)3 / ethanol / Ambient temperature 2: 91 percent / H2, cc.H2SO4 / Pd/C / acetic acid / 25 - 30 °C / 760 Torr View Scheme
参考文献
Tetrahedron Letters, , vol. 25, # 11 p. 1143 - 1146
反应条件
1: 84 percent / pyridine / CH2Cl2 / 0 °C 2: N(C2H5)3 / CH2Cl2 / Ambient temperature 3: H2 / Pd/C / ethanol / 760 Torr / Ambient temperature View Scheme
参考文献
Tetrahedron Letters, , vol. 25, # 11 p. 1143 - 1146
反应条件
1: HCl 2: pyridine / CH2Cl2 / Ambient temperature 3: N(C2H5)3 / CH2Cl2 / Ambient temperature 4: H2 / Pd/C / ethanol / 760 Torr / Ambient temperature View Scheme
参考文献
Tetrahedron Letters, , vol. 25, # 11 p. 1143 - 1146
反应条件
1: pyridine / CH2Cl2 / Ambient temperature 2: N(C2H5)3 / CH2Cl2 / Ambient temperature 3: H2 / Pd/C / ethanol / 760 Torr / Ambient temperature View Scheme
参考文献
Tetrahedron Letters, , vol. 25, # 11 p. 1143 - 1146
反应条件
1: N(C2H5)3 / CH2Cl2 / Ambient temperature 2: H2 / Pd/C / ethanol / 760 Torr / Ambient temperature View Scheme
参考文献
Tetrahedron Letters, , vol. 25, # 11 p. 1143 - 1146
反应条件
1: N(C2H5)3 / CH2Cl2 / Ambient temperature 2: H2 / Pd/C / ethanol / 760 Torr / Ambient temperature View Scheme
参考文献
Tetrahedron Letters, , vol. 25, # 11 p. 1143 - 1146
