7-溴-1,2,4-噻唑并[4,3-a]吡啶合成路线 (共 2 条)
参考文献
3-V BIOSCIENCES, INC.; OSLOB, Johan D.; MCDOWELL, Robert S.; JOHNSON, Russell; YANG, Hanbiao; EVANCHIK, Marc; ZAHARIA, Cristiana A.; CAI, Haiying; HU, Lily W.
Patent: WO2014/8197 A1, 2014 ;
Location in patent: Page/Page column 110 ;
反应条件
1: pyridine; hydrazine / 2 h / 70 °C 2: 100 °C View Scheme