1,5,6,8-四氢-螺[[1]苯并噻吩并[2,3-d]嘧啶-7(4H),2'-[1,3]二氧戊环]-4-酮合成路线 (共 2 条)
反应条件
in formamide
T=140°C; 16 h;
参考文献
BAYER PHARMACEUTICALS CORPORATION
Patent: WO2005/10008 A1, 2005 ;
Location in patent: Page/Page column 125 ;
反应条件
ammonium formate
T=140°C; 16 h;
参考文献
BAYER PHARMACEUTICALS CORPORATION
Patent: WO2006/44524 A1, 2006 ;
Location in patent: Page/Page column 62 ;
WO 2006/044524 A1