反应条件
1: 1.) NaOMe / 1.) THF, -5 deg C, 30 min, 2.) THF, RT, overnight
2: NaOAc / acetic acid / Ambient temperature
View Scheme
参考文献
Kumar, Virendra; Bell, Malcolm R.; Wetzel, Joseph R.; Herrmann, John L.; McGarry, Ruthan; et al.
Journal of Medicinal Chemistry, 1993 , vol. 36, # 22 p. 3278 - 3285