N-(2-二甲基氨基乙基)-3-(4,4,5,5-四甲基-1,3,2-二噁硼烷-2-基)苯甲酰胺合成路线 (共 1 条)
反应条件
benzotriazol-1-ol; 1-ethyl-(3-(3-dimethylamino)propyl)-carbodiimide hydrochloride in N,N-dimethyl-formamide T=20°C; 3 h;
参考文献
Almirall, S.A.
Patent: EP2394998 A1, 2011 ;
Location in patent: Page/Page column 22 ;
EP 2394998 A1