6-氟-1-(2-氟乙基)-7-(4-甲基哌嗪-1-基)-4-氧代-1,8-萘啶-3-羧酸合成路线 (共 3 条)
反应条件
formic acid in water
T=120 - 125°C; 17 h;
参考文献
Matsumoto; Miyamoto; Minamida; Nishimura; Egawa
Journal of Medicinal Chemistry, 1984 , vol. 27, # 3 p. 292 - 301
反应条件
formic acid in ammonium hydroxide
参考文献
Dainippon Pharmaceutical Co., Ltd.; Laboratoire Roger Bellon
Patent: US4496566 A1, 1985 ;
参考文献
Dainippon Pharmaceutical Co., Ltd.; Laboratoire Roger Bellon
Patent: US4496566 A1, 1985 ;