反应条件
1: 1.) thionyl chloride, 2.) NH3 / 2.) ether, 0 deg C, 20-30 min
2: 68 percent / trifluoroacetic anhydride, pyridine / dioxane / 10 °C
View Scheme
参考文献
Adcock, William; Abeywickrema, Anil N.; Kok, Gaik B.
Journal of Organic Chemistry, 1984 , vol. 49, p. 1387 - 1397