1: 95 percent / NEt3; CuI / methanol / 4 h / Heating
2: 87 percent / pyridine / CH2Cl2
3: 49 percent / NH3 / methanol; tetrahydrofuran / 22 h / 50 °C
View Scheme
参考文献
Berry, David A.; Jung, Kee-Yong; Wise, Dean S.; Sercel, Anthony D.; Pearson, William H.; Mackie, Hugh; Randolph, John B.; Somers, Robert L.
Tetrahedron Letters, 2004 , vol. 45, # 11 p. 2457 - 2461
copper(l) iodide; triethylamine in methanol
Robins and Barr method; 4 h; Heating;
参考文献
Berry, David A.; Jung, Kee-Yong; Wise, Dean S.; Sercel, Anthony D.; Pearson, William H.; Mackie, Hugh; Randolph, John B.; Somers, Robert L.
Tetrahedron Letters, 2004 , vol. 45, # 11 p. 2457 - 2461
