potassium hydroxide; tris-(dibenzylideneacetone)dipalladium(0); 2-(dicyclohexylphosphino)-2',4',6'-tri-i-propyl-1,1’-biphenyl in 1,4-dioxane; water
T=100°C; 2 h;
参考文献
SGX PHARMACEUTICALS, INC.
Patent: WO2008/51808 A2, 2008 ;
Location in patent: Page/Page column 84 ;
WO 2008/051808 A2