1-(甲苯-4-磺酰基)-5-乙烯基-1H-吡咯并[2,3-b]吡啶合成路线 (共 1 条)
反应条件
potassium carbonate; tetrakis(triphenylphosphine) palladium(0) in ethylene glycol dimethyl ether; water
T=130°C; 0.166667 h; Microwave;
参考文献
VERTEX PHARMACEUTICALS INCORPORATED
Patent: WO2005/28475 A2, 2005 ;
Location in patent: Page/Page column 216-217 ;
WO 2005/028475 A2