2-氯-5-氟吡啶-3-甲醛合成路线 (共 1 条)
反应条件
1: With hydroxylamine hydrochloride in ethanol; water T=20°C; 1 h; 2: With 1,1'-carbonyldiimidazole in dichloromethane 1 h; Inert atmosphereReflux;
参考文献
ARENA PHARMACEUTICALS, INC.; JONES, Robert M.; BUZARD, Daniel J.; HAN, Sangdon; KIM, Sun Hee; LEHMANN, Juerg; ZHU, Xiuwen
Patent: WO2013/55910 A1, 2013 ;
Location in patent: Page/Page column 106; 107 ;