(2S,4r)-4-氟吡咯烷-2-羧酰胺合成路线 (共 1 条)
反应条件
1: With hydrogenchloride in ethanol
T=20 - 55°C; 62 h;
2: With ammonia in methanol; water
T=20°C; 36 h;
参考文献
Novartis AG
Patent: US2009/163469 A1, 2009 ;
Location in patent: Page/Page column 38 ;
US 20090163469 A1