2,6-二氯-3-甲基苯硼酸合成路线 (共 1 条)
反应条件
1: With n-butyllithium in tetrahydrofuran T=-70°C; 0.5 h; 2: With boric acid trimethyl ester in tetrahydrofuran T=-75 - 20°C; 3: With hydrogenchloride in tetrahydrofuran; water T=0 - 20°C; 2 h;
参考文献
WO2005/44007 A1, ;
Page/Page column 54-55 ;