3-氟-5-(三氟甲基)-2-吡啶羧酰胺合成路线 (共 2 条)
反应条件
sulfuric acid T=105°C; 2 h;
参考文献
MERCK SHARP and DOHME LIMITED
Patent: WO2005/47279 A1, 2005 ;
Location in patent: Page/Page column 57 ;
WO 2005/047279 A1
反应条件
potassium hydroxide; water; bromine T=0 - 20°C; 122 h;
参考文献
MERCK SHARP and DOHME LIMITED
Patent: WO2005/47279 A1, 2005 ;
Location in patent: Page/Page column 57 ;
WO 2005/047279 A1