(5-溴-3-苯并[B]噻吩)甲醇合成路线 (共 1 条)
反应条件
1: With triethylamine; isobutyl chloroformate in tetrahydrofuran T=0°C; 2 h; 2: With sodium tetrahydroborate; water in tetrahydrofuran T=0 - 20°C; 14.5 h;
参考文献
WO2008/109333 A1, ;
Page/Page column 79-80 ;
WO 2008/109333 A1