4-(4,6-二氯-吡啶-2-基)吗啉合成路线 (共 2 条)
反应条件
N-ethyl-N,N-diisopropylamine in 1,4-dioxane
T=85°C; 5 h;
参考文献
SYNTA PHARMACEUTICALS, CORP.
Patent: WO2005/46603 A2, 2005 ;
Location in patent: Page/Page column 85-86 ;
反应条件
sodium carbonate in acetonitrile
T=70°C; 16 h;
参考文献
H. LUNDBECK A/S
Patent: WO2006/92143 A1, 2006 ;
Location in patent: Page/Page column 39 ;
WO 2006/092143 A1