反应条件
sodium hydride
1.) DMF, RT, 0.5 h, 2.) DMF, RT, 20 h; Multistep reaction;
参考文献
Blackburn, Thomas P.; Cox, Barry; Guildford, Allen J.; Count, David J. Le; Middlemiss, Derek N.; et al.
Journal of Medicinal Chemistry, 1987 , vol. 30, # 12 p. 2252 - 2259