3-(N-环丙基氨基磺酰基)苯甲酸合成路线 (共 1 条)
反应条件
1: With triethylamine in tetrahydrofuran
T=0 - 20°C; 3 h;
2: With hydrogenchloride in tetrahydrofuran; water
pH=3;
参考文献
BEIJING HANMI PHARMACEUTICAL CO., LTD.; MA, Long; ZHANG, Bo; LI, Min; XUE, Baoyu; ZHANG, Bi; ZHANG, Wei; QIU, Hongjuan; MOON, Sunghwan; KIM, Maengsup
Patent: WO2012/171488 A1, 2012 ;
Location in patent: Page/Page column 19-20 ;