反应条件
1: 9-methoxy-2,3-dimethyl-9-phenyl-7H-8,9-dihydropyrano[2,3-c]imidazo[1,2-a]pyridine-6-carboxylic acid With O-(benzotriazol-1-yl)-N,N,N',N'-tetramethyluronium tetrafluoroborate in dichloromethane 2 h; Heating; 2: trimethylene imine in dichloromethane T=20°C; 2 h; Further stages. Title compound not separated from byproducts.;
参考文献
Tetrahedron Asymmetry, , vol. 19, # 11 p. 1310 - 1327