1: With sodium carbonate; tetrakis(triphenylphosphine) palladium(0) in water; acetonitrile
T=20 - 90°C; 22 h;
2: With hydrogenchloride in water; acetonitrile
参考文献
GLAXO GROUP LIMITED
Patent: WO2005/58837 A1, 2005 ;
Location in patent: Page/Page column 16 ;
WO 2005/058837 A1
