5-(二氟甲氧基)-1H-吲唑-3-羧酸合成路线 (共 2 条)
反应条件
1: With sodium hydroxide; water
T=60°C; 24 h;
2: With hydrogenchloride
pH=1;
参考文献
MEMORY PHARMACEUTICALS CORPORATION
Patent: WO2006/69097 A2, 2006 ;
Location in patent: Page/Page column 39 ;
WO 2006/069097 A2
反应条件
sodium hydroxide; water
T=60°C; 24 h;
参考文献
MEMORY PHARMACEUTICALS CORPORATION
Patent: WO2005/111038 A2, 2005 ;
Location in patent: Page/Page column 70-72 ;
WO 2005/111038 A2