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1: (naphth-1-yl)acetic acid With lithium diisopropyl amide in tetrahydrofuran T=-78 - 0°C; 2: methyl iodide in tetrahydrofuran T=20°C; Further stages.;
参考文献
Thompson, Hugh W.; Rashid, Shaker Y.
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THE GOVERNMENT OF THE UNITED STATES OF AMERICA AS REPRESENTED BY THE SECRETARY OF THE DEPARTMENT OF HEALTH AND HUMAN SERVICES
Patent: WO2008/22038 A1, 2008 ;
Location in patent: Page/Page column 39-40 ;
WO 2008/022038 A1